1202044-20-9

  • Product Name:Mk 2866
  • Molecular Formula:C19H14F3N3O3
  • Molecular Weight:393.302
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Product Details

pd_meltingpoint:70–74 °C (158–165 °F)

Purity:99%

Mk 2866 1202044-20-9 Powder For Sale with Fast Delivery

  • Molecular Formula:C19H14F3N3O3
  • Molecular Weight:393.302
  • Melting Point:70–74 °C (158–165 °F) 
  • Boiling Point:632.261 °C at 760 mmHg 
  • Flash Point:336.18 °C 
  • PSA:106.14000 
  • Density:1.418 g/cm3 
  • LogP:3.29026 

Ostarine(MK-2866)(Cas 1202044-20-9) Usage

Use

Ostarine, also known as?ostarine MK-2866,?is an investigational?selective androgen receptor modulator?(SARM) developed by?GTx, Inc.?for the treatment of conditions such as?muscle wasting?and?osteoporosis. (2S)-3-(4-Cyanophenoxy-2,3,5,6-d4)-N-[4-cyano-3-(trifluoromethyl)phenyl]-2-hydroxy-2-methylpropanamide is a metabolites of selective androgen receptor modulators (SARM).

Mechanism

Ostarine(MK-2866) attaches to proteins in the body known as androgen receptors. When ostarine binds to these receptors, it tells the muscles in the body to grow. Unlike some other chemicals that bind to androgen receptors, such as?steroids, ostarine doesn't seem to cause as many side effects in other parts of the body.

Health effects

The FDA have warned that SARMs can have serious side effects ranging from risk of heart attack to stroke and liver damage.

Description

Ostarine is an investigational drug that has not yet been approved by the US Food and Drug Administration (FDA). It is part of a class of drugs called selective androgen receptor modulators (SARMs).

InChI:InChI=1/C19H14F3N3O3/c1-18(27,11-28-15-6-2-12(9-23)3-7-15)17(26)25-14-5-4-13(10-24)16(8-14)19(20,21)22/h2-8,27H,11H2,1H3,(H,25,26)/t18-/m1/s1

1202044-20-9 Relevant articles

METABOLITES OF SELECTIVE ANDROGEN RECEPTOR MODULATORS AND METHODS OF USE THEREOF

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Page/Page column 123, (2010/01/12)

This invention provides metabolites of S...

1202044-20-9 Process route

4-cyanophenol-d4
1025089-21-7

4-cyanophenol-d4

(2R)-3-bromo-N-[4-cyano-3-(trifluoromethyl)phenyl]-2-hydroxy-2-methylpropanamide
206193-17-1

(2R)-3-bromo-N-[4-cyano-3-(trifluoromethyl)phenyl]-2-hydroxy-2-methylpropanamide

(S)-N-(4-cyano-3-(trifluoromethyl)phenyl)-3-(4-cyanophenoxy)-2-hydroxy-2-methylpropanamide-d4
1202044-20-9

(S)-N-(4-cyano-3-(trifluoromethyl)phenyl)-3-(4-cyanophenoxy)-2-hydroxy-2-methylpropanamide-d4

Conditions
Conditions Yield
With sodium carbonate; In acetone; for 3h; Reflux;
59.9%

1202044-20-9 Upstream products

  • 1025089-21-7
    1025089-21-7

    4-cyanophenol-d4

  • 206193-17-1
    206193-17-1

    (2R)-3-bromo-N-[4-cyano-3-(trifluoromethyl)phenyl]-2-hydroxy-2-methylpropanamide

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